Brief Information of the Compound and Protein
Compound Name
2-[4-(1H-indazol-5-yloxy)piperidin-1-yl]-3-methyl-6,7-dihydropyrrolo[3,4-b]pyridin-5-one
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PubChem ID
CID: 129277684
Canonical SMILES
Cc1cc2C(=O)NCc2nc1N1CCC(CC1)Oc1ccc2[nH]ncc2c1
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Compound Formula C20H21N5O2
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 14 nM
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