Brief Information of the Compound and Protein
Compound Name
7-[4-(1,3-dihydro-2-benzofuran-5-yloxy)piperidin-1-yl]-6-methyl-2H-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
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PubChem ID
CID: 135154593
Canonical SMILES
Cc1cn2c(n[nH]c2=O)nc1N1CCC(CC1)Oc1ccc2COCc2c1
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Compound Formula C19H21N5O3
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 20 nM
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