Brief Information of the Compound and Protein
Compound Name
1-[(3,4-difluorophenyl)methyl]-N-[[6-(3,3-difluoropyrrolidin-1-yl)pyridin-3-yl]methyl]pyrazole-3-carboxamide
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PubChem ID
CID: 145967526
Canonical SMILES
Fc1ccc(Cn2ccc(n2)C(=O)NCc2ccc(nc2)N2CCC(F)(F)C2)cc1F
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Compound Formula C21H19F4N5O
Compound Structure
Protein Name
Voltage-dependent T-type calcium channel subunit alpha-1H
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated calcium channel
Uniprot ID
O95180
Gene Name
CACNA1H
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 30 nM
   TI
   LI
   LO
   TS