Brief Information of the Compound and Protein
Compound Name
2-ethyl-6,8-dimethyl-3-[[4-[(E)-3-(4-propan-2-ylpiperazin-1-yl)prop-1-enyl]phenyl]methyl]imidazo[1,2-b]pyridazine
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PubChem ID
CID: 145975612
Canonical SMILES
CCc1nc2c(C)cc(C)nn2c1Cc1ccc(\C=C\CN2CCN(CC2)C(C)C)cc1
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Compound Formula C27H37N5
Compound Structure
Protein Name
G-protein coupled receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
P46093
Gene Name
GPR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000017 HeLa Homo sapiens (Human)  1
1
IC50 = 74 nM
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