Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[3,5-difluoro-4-(methanesulfonamido)phenyl]-N-[[2-(4-methylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl]methyl]propanamide
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 PubChem ID
CID: 145960801
Canonical SMILES
CC(C(=O)NCc1ccc(nc1N1CCC(C)CC1)C(F)(F)F)c1cc(F)c(NS(C)(=O)=O)c(F)c1
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Compound Formula C23H27F5N4O3S
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  3
1
IC50 = 8.1 nM
   TI
   LI
   LO
   TS
2
IC50 = 8.7 nM
   TI
   LI
   LO
   TS
3
Ki = 0.2 nM
   TI
   LI
   LO
   TS