Brief Information of the Compound and Protein
Compound Name
(R)-4,6-dimethyl-3-(3-methyl-2-(1-(1-(pyridin-2-ylmethyl)piperidin-4-yl)propyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridine-5-carbonyl)pyridin-2(1H)-one
    Show/Hide
PubChem ID
CID: 145960363
Canonical SMILES
CC[C@@H](c1sc2c(c1C)CN(C(=O)c1c(C)cc(C)[nH]c1=O)CC2)C1CCN(Cc2ccccn2)CC1
    Show/Hide
Compound Formula C30H38N4O2S
Compound Structure
Protein Name
Histone-lysine N-methyltransferase EZH2
Protein Classification
Epigenetic regulator
>
Writer
>
Protein methyltransferase
Uniprot ID
Q15910
Gene Name
EZH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 <= 10 nM
   TI
   LI
   LO
   TS