Brief Information of the Compound and Protein
Compound Name
(R)-3-((2-(1-(1-((2-methoxypyridin-4-yl)methyl)piperidin-4-yl)propyl)-3-methyl-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)methyl)-4,6-dimethylpyridin-2(1H)-one
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PubChem ID
CID: 145961989
Canonical SMILES
CC[C@@H](c1sc2c(c1C)CN(Cc1c(C)cc(C)[nH]c1=O)CC2)C1CCN(Cc2ccnc(OC)c2)CC1
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Compound Formula C31H42N4O2S
Compound Structure
Protein Name
Histone-lysine N-methyltransferase EZH2
Protein Classification
Epigenetic regulator
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Writer
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Protein methyltransferase
Uniprot ID
Q15910
Gene Name
EZH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 <= 10 nM
   TI
   LI
   LO
   TS