Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-N-[4-[4-[(1R,2R,4S)-2-bicyclo[2.2.1]heptanyl]piperazin-1-yl]-3-chlorophenyl]-1-(2-chloro-7-methylthieno[3,2-d]pyrimidin-4-yl)-1,2,4-triazole-3,5-diamine
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 PubChem ID
CID: 137638386
Canonical SMILES
Cc1csc2c(nc(Cl)nc12)-n1nc(Nc2ccc(N3CCN(CC3)[C@@H]3C[C@H]4CC[C@@H]3C4)c(Cl)c2)nc1N
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Compound Formula C26H29Cl2N9S
Compound Structure
Protein Name
 Protein Info 
Tyrosine-protein kinase receptor UFO
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase Axl family
Uniprot ID
P30530
Gene Name
AXL
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000017 HeLa
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 216 nM
   TI
   LI
   LO
   TS