Brief Information of the Compound and Protein
Compound Name
N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]propane-2-sulfonamide
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PubChem ID
CID: 45380469
SID: 93372122
Canonical SMILES
CC(C)S(=O)(=O)Nc1cccc(c1)[C@@H](O)CNCCOc1ccc2c(C)n[nH]c2c1
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Compound Formula C21H28N4O4S
Compound Structure
Protein Name
Alpha-1A adrenergic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Adrenergic receptor
Uniprot ID
P35348
Gene Name
ADRA1A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 1757 nM
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