Brief Information of the Compound and Protein
Compound Name
N-[(2,6-difluorophenyl)methyl]-3-(9-oxa-3,4,6,12-tetrazatricyclo[8.4.0.02,6]tetradeca-1(10),2,4,11,13-pentaen-5-ylmethylamino)benzamide
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PubChem ID
CID: 137640915
Canonical SMILES
Fc1cccc(F)c1CNC(=O)c1cccc(NCc2nnc3-c4ccncc4OCCn23)c1
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Compound Formula C24H20F2N6O2
Compound Structure
Protein Name
Beta-adrenergic receptor kinase 1
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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AGC protein kinase group
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AGC protein kinase GRK family
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AGC protein kinase BARK subfamily
Uniprot ID
P25098
Gene Name
GRK2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 23000 nM
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