Brief Information of the Compound and Protein
Compound Name
3-(9-oxa-3,4,6,12-tetrazatricyclo[8.4.0.02,6]tetradeca-1(10),2,4,11,13-pentaen-5-ylmethylamino)-N-[[2-(trifluoromethyl)phenyl]methyl]benzamide
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PubChem ID
CID: 137638433
Canonical SMILES
FC(F)(F)c1ccccc1CNC(=O)c1cccc(NCc2nnc3-c4ccncc4OCCn23)c1
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Compound Formula C25H21F3N6O2
Compound Structure
Protein Name
Rhodopsin kinase GRK1
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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AGC protein kinase group
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AGC protein kinase GRK family
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AGC protein kinase GRK subfamily
Uniprot ID
Q15835
Gene Name
GRK1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 270 nM
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