Brief Information of the Compound and Protein
Compound Name
2-(6-cyclopropyl-5,7-dioxo-3,4-dihydro-2H-pyrrolo[3,4-b]pyridin-1-yl)-N-[6-(5-fluoropyridin-3-yl)pyridazin-3-yl]acetamide
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PubChem ID
CID: 118174232
Canonical SMILES
Fc1cncc(c1)-c1ccc(NC(=O)CN2CCCC3=C2C(=O)N(C2CC2)C3=O)nn1
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Compound Formula C21H19FN6O3
Compound Structure
Protein Name
Protein-serine O-palmitoleoyltransferase porcupine
Protein Classification
Enzyme
>
Transferase
Uniprot ID
Q9H237
Gene Name
PORCN
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 11 nM
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