Brief Information of the Compound and Protein
Compound Name
1-[5-fluoro-4-(3-fluorophenyl)-2-methoxyphenyl]-N-(1,2-oxazol-3-yl)-2-oxoquinazoline-6-sulfonamide
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PubChem ID
CID: 137638107
Canonical SMILES
COc1cc(c(F)cc1-n1c2ccc(cc2cnc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
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Compound Formula C24H16F2N4O5S
Compound Structure
Protein Name
Sodium channel protein type 9 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q15858
Gene Name
SCN9A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1800 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 1750 nM