Brief Information of the Compound and Protein
Compound Name
1-[6-[(2R)-4-[1-[[3-(2-methoxyethoxy)phenyl]methyl]-3-methylthieno[2,3-c]pyrazole-5-carbonyl]-2-methylpiperazin-1-yl]pyridin-3-yl]ethanone
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PubChem ID
CID: 137655175
Canonical SMILES
COCCOc1cccc(Cn2nc(C)c3cc(sc23)C(=O)N2CCN([C@H](C)C2)c2ccc(cn2)C(C)=O)c1
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Compound Formula C29H33N5O4S
Compound Structure
Protein Name
Steroid hormone receptor ERR1
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 3
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Nuclear hormone receptor subfamily 3 group B
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Nuclear hormone receptor subfamily 3 group B member 1
Uniprot ID
P11474
Gene Name
ESRRA
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 22 nM
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