Brief Information of the Compound and Protein
Compound Name
4-[2-(3,5-dimethylpyrazol-1-yl)ethoxy]-3-methyl-1-(7H-purin-6-yl)-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one
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PubChem ID
CID: 137649835
Canonical SMILES
Cc1cc(C)n(CCOC2CC(=O)Nc3c2c(C)nn3-c2ncnc3nc[nH]c23)n1
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Compound Formula C19H21N9O2
Compound Structure
Protein Name
G-protein coupled receptor 39
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
O43194
Gene Name
GPR39
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 16 nM
   TI
   LI
   LO
   TS
2
EC50 = 2004 nM
   TI
   LI
   LO
   TS