Brief Information of the Compound and Protein
Compound Name
US9452986, 521
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PubChem ID
CID: 118273365
Canonical SMILES
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CCNC(=O)C2)nc1
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Compound Formula C21H17F3N4O3
Compound Structure
Protein Name
Sodium channel protein type 10 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q9Y5Y9
Gene Name
SCN10A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1100 nM
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