Brief Information of the Compound and Protein
Compound Name
US9447114, 26
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PubChem ID
CID: 118863119
Canonical SMILES
Cn1c2sc(c(Cc3ccc(Cl)cc3)c2c(=O)n(CCCO)c1=O)-c1cccc(OC(F)(F)F)c1
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Compound Formula C24H20ClF3N2O4S
Compound Structure
Protein Name
Short transient receptor potential channel 5
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9UL62
Gene Name
TRPC5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000058 T-REx-293 Homo sapiens (Human)  2
1
IC50 < 1 nM
   TI
   LI
   LO
   TS
2
IC50 = 1.91 nM
   TI
   LI
   LO
   TS