Brief Information of the Compound and Protein
Compound Name
 Compound Info 
US9394293, G159a
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 PubChem ID
CID: 71609694
Canonical SMILES
Cc1ccc2nc(NC(=O)c3ccc(cc3)-c3ncc(C[C@@H](O)CO)cc3F)sc2c1
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Compound Formula C23H20FN3O3S
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000650 CHO-hTRPV1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 29.6 nM
   TI
   LI
   LO
   TS
2
IC50 = 879 nM
   TI
   LI
   LO
   TS