Brief Information of the Compound and Protein
Compound Name
 Compound Info 
US9394293, G158a
    Show/Hide
 PubChem ID
CID: 71609695
Canonical SMILES
OC[C@H](O)Cc1cnc(c(F)c1)-c1ccc(cc1)C(=O)Nc1nc2ccc(F)cc2s1
    Show/Hide
Compound Formula C22H17F2N3O3S
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000650 CHO-hTRPV1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 77 nM
   TI
   LI
   LO
   TS
2
IC50 = 598 nM
   TI
   LI
   LO
   TS