Brief Information of the Compound and Protein
Compound Name
US9394293, G215a
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PubChem ID
CID: 71609697
Canonical SMILES
Cc1cc2nc(NC(=O)c3ccc(cc3)-c3ncc(C[C@@H](O)CO)cc3F)sc2cc1C
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Compound Formula C24H22FN3O3S
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000650 CHO-hTRPV1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 219 nM
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