Brief Information of the Compound and Protein
Compound Name
US9340500, I-029
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PubChem ID
CID: 89946659
Canonical SMILES
CC(C)c1cccc(NC(=O)c2cc(-c3ccccc3)n(CCCN3CCOCC3)c2C)c1
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Compound Formula C28H35N3O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9HBA0
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL001031 hTRPV4/CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 519 nM
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   LI
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