Brief Information of the Compound and Protein
Compound Name
US9340500, I-082
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PubChem ID
CID: 71465983
SID: 163428519
Canonical SMILES
Cc1c(NC(=O)c2cccc(c2)C(F)(F)F)cc(-c2ccccc2)n1CCCN1CCOCC1
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Compound Formula C26H28F3N3O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9HBA0
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL001031 hTRPV4/CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1437 nM
   TI
   LI
   LO
   TS