Brief Information of the Compound and Protein
Compound Name
US9212171, 29
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PubChem ID
CID: 70937838
Canonical SMILES
CN1[C@H]2CCC[C@H]2[C@@H](C1=O)c1ccc(cn1)C#Cc1ccc(F)cc1
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Compound Formula C21H19FN2O
Compound Structure
Protein Name
Metabotropic glutamate receptor 5
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
P41594
Gene Name
GRM5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 78 nM
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