Brief Information of the Compound and Protein
Compound Name
US9273043, B155(h)
    Show/Hide
PubChem ID
CID: 117678419
Canonical SMILES
C[C@H](O)[C@@H](O)c1cnc(N2CCN([C@@H](C)C2)C(=O)Nc2nc3cc(F)ccc3s2)c(F)c1
    Show/Hide
Compound Formula C21H23F2N5O3S
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000650 CHO-hTRPV1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 107 nM
   TI
   LI
   LO
   TS