Brief Information of the Compound and Protein
Compound Name
4-[5-(dimethylcarbamoyl)-3-(2,4,6-trimethylphenyl)sulfanylindazol-1-yl]benzoic acid
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PubChem ID
CID: 134131811
Canonical SMILES
CN(C)C(=O)c1ccc2n(nc(Sc3c(C)cc(C)cc3C)c2c1)-c1ccc(cc1)C(O)=O
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Compound Formula C26H25N3O3S
Compound Structure
Protein Name
Nuclear receptor ROR-gamma
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group F
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Nuclear hormone receptor subfamily 1 group F member 3
Uniprot ID
P51449
Gene Name
RORC
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000789 HG5LN Homo sapiens (Human)  1
1
IC50 = 2700 nM
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