Brief Information of the Compound and Protein
Compound Name
(5S)-5-amino-21-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,7,16,18,24-pentazatricyclo[15.5.2.020,23]tetracosa-17,19,21,23-tetraen-6-one
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PubChem ID
CID: 134151512
Canonical SMILES
CN1CCN(Cc2ccc(cc2)-c2cn3CCC[C@H](N)C(=O)NCCCCCCCCNc4ncc2c3n4)CC1
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Compound Formula C31H46N8O
Compound Structure
Protein Name
Tyrosine-protein kinase Mer
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase Axl family
Uniprot ID
Q12866
Gene Name
MERTK
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 30 nM