Brief Information of the Compound and Protein
Compound Name
 Compound Info 
18-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1,13,15,21-tetrazatricyclo[12.5.2.017,20]henicosa-14,16,18,20-tetraen-5-ol
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 PubChem ID
CID: 134132904
Canonical SMILES
CN1CCN(Cc2ccc(cc2)-c2cn3CCCC(O)CCCCCCCNc4ncc2c3n4)CC1
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Compound Formula C29H42N6O
Compound Structure
Protein Name
 Protein Info 
Tyrosine-protein kinase Mer
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase Axl family
Uniprot ID
Q12866
Gene Name
MERTK
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 43 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 1.8 nM