Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(+/-)-N-Benzyl-3,5-dimethyl-1-(phenylmethyl-d2)-1,2,3,5-tetrahydro-4H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
    Show/Hide
 PubChem ID
CID: 134156616
Canonical SMILES
[2H]C([2H])(c1ccccc1)N1C[C@@H](C)N(C(=O)NCc2ccccc2)[C@@H](C)c2ccncc21
    Show/Hide
Compound Formula C25H28N4O
Compound Structure
Protein Name
 Protein Info 
Voltage-dependent T-type calcium channel subunit alpha-1H
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Voltage-gated calcium channel
Uniprot ID
O95180
Gene Name
CACNA1H
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 230 nM
   TI
   LI
   LO
   TS