Brief Information of the Compound and Protein
Compound Name
N-(4-bromophenyl)-5-(2-hydroxyethyl)-5-(4-methoxyphenyl)-3-pyridin-3-yl-4H-pyrazole-1-carboxamide
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PubChem ID
CID: 134133525
Canonical SMILES
COc1ccc(cc1)C1(CCO)CC(=NN1C(=O)Nc1ccc(Br)cc1)c1cccnc1
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Compound Formula C24H23BrN4O3
Compound Structure
Protein Name
Voltage-dependent T-type calcium channel subunit alpha-1H
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated calcium channel
Uniprot ID
O95180
Gene Name
CACNA1H
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 140 nM
   TI
   LI
   LO
   TS