Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-[[3-chloro-4-[2-[6-(2H-tetrazol-5-yl)pyridin-3-yl]cyclopropyl]phenoxy]methyl]-5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazole
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 PubChem ID
CID: 50943000
SID: 115948797
Canonical SMILES
Clc1cccc(Cl)c1-c1noc(C2CC2)c1COc1ccc(C2CC2c2ccc(nc2)-c2nnn[nH]2)c(Cl)c1
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Compound Formula C28H21Cl3N6O2
Compound Structure
Protein Name
 Protein Info 
Bile acid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
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Nuclear hormone receptor subfamily 1
>
Nuclear hormone receptor subfamily 1 group H
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Nuclear hormone receptor subfamily 1 group H member 4
Uniprot ID
Q96RI1
Gene Name
NR1H4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 111 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 131 nM