Brief Information of the Compound and Protein
Compound Name
(3aS,6aS)-5-[1-(2-fluorophenyl)indazol-4-yl]-1-(3-hydroxy-3-methylbutanoyl)-3,3a,4,6a-tetrahydro-2H-pyrrolo[2,3-c]pyrrol-6-one
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PubChem ID
CID: 122513481
Canonical SMILES
CC(C)(O)CC(=O)N1CC[C@H]2CN(C(=O)[C@@H]12)c1cccc2n(ncc12)-c1ccccc1F
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Compound Formula C24H25FN4O3
Compound Structure
Protein Name
Sodium channel protein type 9 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q15858
Gene Name
SCN9A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000131 HEK293-F Homo sapiens (Human)  1
1
IC50 = 1350 nM
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