Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(3aR,6aS)-5-[1-(2-fluorophenyl)indazol-4-yl]-2-(3-hydroxy-3-methylbutanoyl)-3,3a,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-4-one
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 PubChem ID
CID: 122513516
Canonical SMILES
CC(C)(O)CC(=O)N1C[C@H]2CN(C(=O)[C@H]2C1)c1cccc2n(ncc12)-c1ccccc1F
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Compound Formula C24H25FN4O3
Compound Structure
Protein Name
 Protein Info 
Sodium channel protein type 9 subunit alpha
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q15858
Gene Name
SCN9A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000131 HEK293-F
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 340 nM
   TI
   LI
   LO
   TS
2
IC50 = 3900 nM
   TI
   LI
   LO
   TS