Brief Information of the Compound and Protein
Compound Name
[(3S)-3-hydroxypyrrolidin-1-yl]-[3-[(1-methylindazol-5-yl)methyl]-2H-indazol-5-yl]methanone
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PubChem ID
CID: 118960086
Canonical SMILES
Cn1ncc2cc(Cc3n[nH]c4ccc(cc34)C(=O)N3CC[C@H](O)C3)ccc12
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Compound Formula C21H21N5O2
Compound Structure
Protein Name
Cyclin-dependent kinase 8
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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CMGC protein kinase group
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CMGC protein kinase CDK family
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CMGC protein kinase CDK8 subfamily
Uniprot ID
P49336
Gene Name
CDK8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 43 nM
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