Brief Information of the Compound and Protein
Compound Name
(3-methoxyazetidin-1-yl)-[3-[(1-methylindazol-5-yl)methyl]-2H-indazol-5-yl]methanone
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PubChem ID
CID: 127034391
Canonical SMILES
COC1CN(C1)C(=O)c1ccc2[nH]nc(Cc3ccc4n(C)ncc4c3)c2c1
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Compound Formula C21H21N5O2
Compound Structure
Protein Name
Cyclin-dependent kinase 8
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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CMGC protein kinase group
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CMGC protein kinase CDK family
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CMGC protein kinase CDK8 subfamily
Uniprot ID
P49336
Gene Name
CDK8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 18 nM
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