Brief Information of the Compound and Protein
Compound Name
4-N-{1-[2-(Biphenyl-2-yloxy)ethyl]piperidin-4-yl}-isoquinolinesulfonamide
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PubChem ID
CID: 127041107
Canonical SMILES
O=S(=O)(NC1CCN(CCOc2ccccc2-c2ccccc2)CC1)c1cncc2ccccc12
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Compound Formula C28H29N3O3S
Compound Structure
Protein Name
5-hydroxytryptamine receptor 1A
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P08908
Gene Name
HTR1A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 74 nM
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   LI
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