Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(benzo[d][1,3]dioxol-5-yl)-2-(4-((2-ethyl-4,6-dimethyl-1H-benzo[d]imidazol-1-yl)methyl)-2-propylphenoxy)-N-(4-isopropylphenylsulfonyl)acetamide
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 PubChem ID
CID: 127034758
Canonical SMILES
CCCc1cc(Cn2c(CC)nc3c(C)cc(C)cc32)ccc1OC(C(=O)NS(=O)(=O)c1ccc(C(C)C)cc1)c1ccc2c(c1)OCO2
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Compound Formula C39H43N3O6S
Compound Structure
Protein Name
 Protein Info 
Endothelin-1 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Endothelin receptor
Uniprot ID
P25101
Gene Name
EDNRA
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 24 nM
   TI
   LI
   LO
   TS