Brief Information of the Compound and Protein
Compound Name
(S)-4-(3-ethoxy-4-oxo-2-(1-(4-(trifluoromethyl)phenyl)ethylamino)-3,4,5,6,7,8-hexahydropyrido[4,3-d]pyrimidine-6-carbonyl)benzonitrile
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PubChem ID
CID: 57378695
SID: 136884591
Canonical SMILES
CCOn1c(N[C@@H](C)c2ccc(C(F)(F)F)cc2)nc2c(c1=O)CN(C(=O)c1ccc(C#N)cc1)CC2
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Compound Formula C26H24F3N5O3
Compound Structure
Protein Name
Prolactin-releasing peptide receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Prolactin-releasing peptide receptor
Uniprot ID
P49683
Gene Name
PRLHR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 156 nM
   TI
   LI
   LO
   TS
2
Ki = 11 nM
   TI
   LI
   LO
   TS