Brief Information of the Compound and Protein
Compound Name
2-Methoxy-6-(6-methoxy-4-((2-phenylpyrimidin-4-yl)methoxy)benzofuran-2-yl)imidazo[2,1-b][1,3,4]thiadiazole
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PubChem ID
CID: 72192130
Canonical SMILES
COc1nn2cc(nc2s1)-c1cc2c(OCc3ccnc(n3)-c3ccccc3)cc(OC)cc2o1
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Compound Formula C25H19N5O4S
Compound Structure
Protein Name
Proteinase-activated receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Protease-activated receptor
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Protease-activated receptor
Uniprot ID
Q96RI0
Gene Name
F2RL3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 0.9 nM
   TI
   LI
   LO
   TS
2
IC50 = 0.92 nM
   TI
   LI
   LO
   TS