Brief Information of the Compound and Protein
Compound Name
US10047103, 186
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PubChem ID
CID: 89879347
Canonical SMILES
CNC(=O)c1ccc(cc1)-c1nc(COc2cc(F)cc3oc(cc23)-c2cn3nc(OC)sc3n2)c(C)s1
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Compound Formula C26H20FN5O4S2
Compound Structure
Protein Name
Proteinase-activated receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Protease-activated receptor
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Protease-activated receptor
Uniprot ID
Q96RI0
Gene Name
F2RL3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 0.58 nM
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   LI
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   TS