Brief Information of the Compound and Protein
Compound Name
US10047103, 250
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PubChem ID
CID: 117981533
Canonical SMILES
COc1cc(OCc2csc(n2)N(C)CCC#N)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
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Compound Formula C24H22N6O3S
Compound Structure
Protein Name
Proteinase-activated receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Protease-activated receptor
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Protease-activated receptor
Uniprot ID
Q96RI0
Gene Name
F2RL3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 3.6 nM
   TI
   LI
   LO
   TS