Brief Information of the Compound and Protein
Compound Name
US8969325, 208
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PubChem ID
CID: 89646648
Canonical SMILES
CN1Cc2ccc(NC(=O)N[C@@H]3CC(C)(C)Oc4nc(ccc34)C(F)(F)F)cc2NC1=O
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Compound Formula C21H22F3N5O3
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1300 nM
   TI
   LI
   LO
   TS