Brief Information of the Compound and Protein
Compound Name
US8853242, 159
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PubChem ID
CID: 50923583
SID: 113917751
Canonical SMILES
COc1cccc(F)c1-c1ncc(F)c2ccc(cc12)C(=O)N=C(N)N
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Compound Formula C18H14F2N4O2
Compound Structure
Protein Name
5-hydroxytryptamine receptor 5A
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P47898
Gene Name
HTR5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 7.1 nM
   TI
   LI
   LO
   TS