Brief Information of the Compound and Protein
Compound Name
US8993765, 12
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PubChem ID
CID: 57524672
SID: 137282343
Canonical SMILES
CC1Cc2c(CN1)c1ccc(nc1n2C)N1CCN(CCc2ccc(F)cc2)CC1=O
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Compound Formula C24H28FN5O
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
Ki = 58 nM
   TI
   LI
   LO
   TS