Brief Information of the Compound and Protein
Compound Name
4-(4-bromo-2-ethylphenyl)-8-[butyl(ethyl)amino]-6-methyl-1,3-dihydropyrido[2,3-b]pyrazin-2-one
    Show/Hide
PubChem ID
CID: 90231885
Canonical SMILES
CCCCN(CC)c1cc(C)nc2N(CC(=O)Nc12)c1ccc(Br)cc1CC
    Show/Hide
Compound Formula C22H29BrN4O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Corticotropin releasing factor receptor
>
Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
Ki = 2.5 nM
   TI
   LI
   LO
   TS