Brief Information of the Compound and Protein
Compound Name
2-[(2-acetyl-3,4-dihydro-1H-isoquinolin-7-yl)oxy]-N-(5-pyrazin-2-ylpyridin-2-yl)acetamide
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PubChem ID
CID: 122192862
Canonical SMILES
CC(=O)N1CCc2ccc(OCC(=O)Nc3ccc(cn3)-c3cnccn3)cc2C1
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Compound Formula C22H21N5O3
Compound Structure
Protein Name
Protein-serine O-palmitoleoyltransferase porcupine
Protein Classification
Enzyme
>
Transferase
Uniprot ID
Q9H237
Gene Name
PORCN
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000575 L Wnt-3A Mus musculus (Mouse)  1
1
IC50 = 24 nM
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