Brief Information of the Compound and Protein
Compound Name
[(1S,2R,4R)-2-[2-[3-(1H-benzimidazol-2-yl)propyl-methylamino]ethyl]-6-fluoro-4-hydroxy-1-propan-2-yl-3,4-dihydro-1H-naphthalen-2-yl] 2-methylpropanoate
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PubChem ID
CID: 122187210
Canonical SMILES
CC(C)[C@H]1c2ccc(F)cc2[C@H](O)C[C@@]1(CCN(C)CCCc1nc2ccccc2[nH]1)OC(=O)C(C)C
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Compound Formula C30H40FN3O3
Compound Structure
Protein Name
Voltage-dependent T-type calcium channel subunit alpha-1H
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated calcium channel
Uniprot ID
O95180
Gene Name
CACNA1H
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 107 nM
   TI
   LI
   LO
   TS