Brief Information of the Compound and Protein
Compound Name
4-[(5-chloropyridin-2-yl)methoxy]-1-[2-[4-[(dimethylamino)methyl]phenyl]-2-oxoethyl]pyridin-2-one
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PubChem ID
CID: 44193451
SID: 85189244
Canonical SMILES
CN(C)Cc1ccc(cc1)C(=O)Cn1ccc(OCc2ccc(Cl)cn2)cc1=O
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Compound Formula C22H22ClN3O3
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000076 CHO/Galpha16 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 41 nM
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