Brief Information of the Compound and Protein
Compound Name
US8933079, 3.9
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PubChem ID
CID: 71731948
Canonical SMILES
CN(C)Cc1ccc(C(=O)Cn2ccc(OCc3ccc(Cl)cn3)cc2=O)c(C)c1
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Compound Formula C23H24ClN3O3
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000076 CHO/Galpha16 Cricetulus griseus (Chinese hamster)  2
1
IC50 = 32 nM
   TI
   LI
   LO
   TS
2
IC50 = 33 nM
   TI
   LI
   LO
   TS