Brief Information of the Compound and Protein
Compound Name
2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2,6-dimethoxyphenyl)methyl]ethanamine
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PubChem ID
CID: 122180973
Canonical SMILES
COc1cccc(OC)c1CNCCc1cc(OC)c(Br)cc1OC
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Compound Formula C19H24BrNO4
Compound Structure
Protein Name
5-hydroxytryptamine receptor 2C
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P28335
Gene Name
HTR2C
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 87096.36 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 17.38 nM