Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(benzo[d][1,3]dioxol-5-ylmethylamino)-5-((1R,5S)-8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)nicotinamide
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 PubChem ID
CID: 122180024
Canonical SMILES
O=C(NC[C@H]1COc2ccccc2O1)c1cc(N2C[C@H]3CC[C@@H](C2)O3)cnc1NCc1ccc2c(c1)OCO2
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Compound Formula C29H30N4O6
Compound Structure
Protein Name
 Protein Info 
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
O08725
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 560 nM
   TI
   LI
   LO
   TS